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Sun, M-K., and Alkon, D.L. (2001) Pharmacological enhancement of synaptic efficacy, spatial learning and memory through carbonic anhydrase activation in rats. Journal of Pharmacology and Experimental Therapeutics 297, 961–967.
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Sun, M.K., Dahl, D., and Alkon, D.L. (2001) Heterosynaptic transformation of GABAergic gating in the hippocampus and effects of carbonic anhydrase inhibition. Journal of Pharmacology and Experimental Therapeutics 296, 811–817.
Supuran, C.T. (1991) Design of carbonic anhydrase inhibitors and activators. Ph. D. Thesis, Polytechnic University, Bucharest, pp. 1–148.
Supuran, C.T. (1992) Carbonic anhydrase activators. Part 4. A general mechanism of action for activators of isozymes I, II and III. Revue Roumaine de Chimie 37, 411–421.
Supuran, C.T., and Balaban, A.T. (1994) Carbonic anhydrase activators. Part 8. pKa-activation relationship in a series of amino acid derivatives activators of isozyme II. Revue Roumaine de Chimie 39, 107–113.
Supuran, C.T., Balaban, A.T., Cabildo, P., Claramunt, R.M., Lavandera, J.L., and Elguero, J. (1993a) Carbonic anhydrase activators. Part 7. Isozyme II activation with bis-azolyl- methanes, -ethanes and related azoles. Biological and Pharmaceutical Bulletin 16, 1236–1239.
Supuran, C.T., Barboiu, M., Luca, C., Pop, E., Brewster, M.E., and Dinculescu, A. (1996a) Carbonic anhydrase activators. Part 14. Synthesis of monoand bis-pyridinium salt derivatives of 2-amino-5-(2-aminoethyl)- and 2-amino-5-(3-aminopropyl)-1,3,4-thi- adiazole, and their interaction with isozyme II. European Journal of Medicinal Chemistry 31, 597–606.
Supuran, C.T., Claramunt, R.M., Lavandera, J.L., and Elguero, J. (1996b) Carbonic anhydrase activators. Part 15. A kinetic study of the interaction of bovine isozyme II with pyrazoles, bisand tris-azolylmethanes. Biological and Pharmaceutical Bulletin 19, 1417–1422.
Supuran, C.T., Dinculescu, A., and Balaban, A.T. (1993b) Carbonic anhydrase activators. Part 5. CA II activation by 2,4,6-trisubstituted pyridinium cations with 1-(-aminoalkyl)side chains. Revue Roumaine de Chimie 38, 343–349.
Supuran, C.T., Dinculescu, A., Manole, G., Savan, F., Puscas, I., and Balaban, A.T. (1991) Carbonic anhydrase activators. Part 2. Amino acids and some of their derivatives may act as potent enzyme activators. Revue Roumaine de Chimie 36, 937–946.
Supuran, C.T., and Puscas, I. (1994) Carbonic anhydrase activators. In Carbonic Anhydrase and Modulation of Physiologic and Pathologic Processes in the Organism, Puscas, I. (Ed.), Helicon, Timisoara, Romania, pp. 113–145.
Supuran, C.T., and Scozzafava, A. (1999) Carbonic anhydrase activators. Part 23. Aminoacyl/dipeptidyl histamine derivatives bind with high affinity to isozymes I, II and IV and act as efficient activators. Bioorganic Medicinal Chemistry 7, 2397–2406.
Supuran, C.T., and Scozzafava, A. (2000a) Activation of carbonic anhydrase isozymes. In The Carbonic Anhydrases — New Horizons, Chegwidden, W.R., Edwards, Y., and Carter, N. (Eds.), Birkhäuser Verlag, Basel, pp. 197–219.
Supuran, C.T., and Scozzafava, A. (2000b) Carbonic anhydrase inhibitors and their therapeutic potential. Expert Opinion on Therapeutic Patents 10, 575–600.
Supuran, C.T., and Scozzafava, A. (2000c) Carbonic anhydrase activators: Synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(arylsulfonylureido-amino acyl)ethyl-1H-imidazole. Journal of Enzyme Inhibition 15, 471–486.
Supuran, C.T., and Scozzafava, A. (2001) Carbonic anhydrase inhibitors. Current Medicinal Chemistry — Immunologic, Endocrine and Metabolic Agents 1, 61–97.